PD158780
Product Specifications
CAS Number
171179-06-9
Target
EGFR
Related Pathways
Angiogenesis, Tyrosine Kinase/Adaptors, JAK/STAT signaling
Purity
0.9916
Bioactivity
PD 158780 reversibly inhibits auto and transphosphorylation of all four members of the ErbB receptor superfamily: EGFR, ErbB2, ErbB3, and ErbB4 (IC50s: 8μM, 49 nM, 52 nM, and 52 nM in cell assay) .
Smiles
CNc1cc2c(Nc3cccc(Br)c3)ncnc2cn1
Molecular Formula
C14H12BrN5
Molecular Weight
330.18
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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