BI-1347
Product Specifications
CAS Number
2163056-91-3
Target
CDK
Related Pathways
Cell Cycle/Checkpoint
Purity
0.9963
Bioactivity
BI-1347 is a potent, selective inhibitor of CDK8/cyclinC (IC50: 1 nM) . It shows tumor growth inhibition in an in vivo xenograft model.
Smiles
CN(C)C(=O)Cn1cc(cn1)-c1ccc(cc1)-c1cncc2ccccc12
Molecular Formula
C22H20N4O
Molecular Weight
356.42
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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