CK1-IN-1
Product Specifications
CAS Number
1784751-20-7
Target
Casein Kinase, p38 MAPK
Related Pathways
MAPK, Stem Cells, Metabolism
Purity
0.9879
Bioactivity
CK1-IN-1 (PUN51207) is a casein kinase 1 (CK1) inhibitor. CK1-IN-1 has IC50s of 15 nM, 16 nM, 73 nM for CK1δ, and CK1ε, p38σ MAPK, respectively.
Smiles
Fc1ccc(cc1)-c1nc([nH]c1-c1ccncc1)-c1ccc2ccccc2c1F
Molecular Formula
C24H15F2N3
Molecular Weight
383.39
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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