Sparsentan
Product Specifications
CAS Number
254740-64-2
Target
RAAS, Endothelin Receptor
Related Pathways
Endocrinology/Hormones, GPCR/G Protein
Purity
0.9881
Bioactivity
Sparsentan (DARA-a) is a first-in-class orally active and highly potent dual endothelin A and angiotensin II receptor antagonist (Ki of 9.3 and 0.8 nM, respectively)
Smiles
CCCCC1=NC2(CCCC2)C(=O)N1Cc1ccc(c(COCC)c1)-c1ccccc1S(=O)(=O)Nc1noc(C)c1C
Molecular Formula
C32H40N4O5S
Molecular Weight
592.75
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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