ERK5-IN-1
Product Specifications
CAS Number
1234479-76-5
Target
ERK
Related Pathways
MAPK
Purity
0.9942
Bioactivity
ERK5-IN-1 is a potent ERK5 inhibitor (IC50: 87 nM) and also inhibits LRRK2[G2019S] (IC50: 26 nM) .
Smiles
COc1cc(ccc1Nc1ncc2N(C)C(=O)c3ccccc3N(C)c2n1)N1CCN(C)CC1
Molecular Formula
C25H29N7O2
Molecular Weight
459.54
Shipping Conditions
Cool pack
Storage Temperature
-20°C
Product Datasheet
https://www.targetmol.com/attachment/DataSheet/34FB8C44-AA7A-4229-8CDD-BB79B6513D2D/T5184
Available Sizes
Curated Selection
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