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ERK5-IN-1

Product Specifications

CAS Number

1234479-76-5

Target

ERK

Related Pathways

MAPK

Purity

0.9942

Bioactivity

ERK5-IN-1 is a potent ERK5 inhibitor (IC50: 87 nM) and also inhibits LRRK2[G2019S] (IC50: 26 nM) .

Smiles

COc1cc(ccc1Nc1ncc2N(C)C(=O)c3ccccc3N(C)c2n1)N1CCN(C)CC1

Molecular Formula

C25H29N7O2

Molecular Weight

459.54

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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