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PF-4800567

Product Specifications

CAS Number

1188296-52-7

Target

Casein Kinase

Related Pathways

Stem Cells, Metabolism

Purity

0.9976

Bioactivity

PF-4800567 is a selective inhibitor of casein kinase 1ε (CK1ε; IC50 = 32 nM) with greater than 20-fold selectivity over CK1δ.

Smiles

Nc1ncnc2n(nc(COc3cccc(Cl)c3)c12)C1CCOCC1

Molecular Formula

C17H18ClN5O2

Molecular Weight

359.81

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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