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PF-01247324

Product Specifications

CAS Number

875051-72-2

Target

Sodium Channel

Related Pathways

Membrane transporter/Ion channel

Purity

0.9994

Bioactivity

PF-01247324 is a selective and orally bioavailable Nav1.8 channel blocker [IC50: 196 nM].

Smiles

CNC(=O)c1ccc(c(N)n1)-c1cc(Cl)cc(Cl)c1Cl

Molecular Formula

C13H10Cl3N3O

Molecular Weight

330.6

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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