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GIBH-130

Product Specifications

CAS Number

1252608-59-5

Target

Interleukin|||IL Receptor|||TNF

Related Pathways

Apoptosis|||Immunology/Inflammation

Purity

0.9986

Bioactivity

GIBH-130 markedly inhibits the IL-1? secretion by activated microglia (IC50: 3.4 nM) . GIBH-130 is an effective inhibitor of neuroinflammation.

Smiles

Cc1cc(nnc1C(=O)N1CCN(CC1)c1ncccn1)-c1ccccc1

Molecular Formula

C20H20N6O

Molecular Weight

360.41

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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