What is the catalog number for ML221?

The catalog number for ML221 is T4390.

What sizes are available for ML221?

ML221 is available in the following size(s): 2 mg, 5 mg, 1 mL - 10 mM (in DMSO), 10 mg, 25 mg, 50 mg, 100 mg, 200 mg.

How many pack sizes does ML221 come in?

ML221 is available in 8 different pack sizes.

ML221 is currently made to order / not held in immediate stock. Contact us for lead time.

Who manufactures ML221?

ML221 is manufactured by Molfinity.

What is the estimated delivery time for ML221?

Estimated delivery time for ML221 is approximately 10 business day(s), depending on your location.

ML221

Product Specifications

CAS Number

877636-42-5

Target

Arrestin, Apelin receptor

Related Pathways

GPCR/G Protein

Purity

0.9774

Bioactivity

ML221 is a potent apelin /APJ functional antagonist, inhibiting apelin-13-mediated activation of APJ, with IC50s of 0.70 μM in the cAMP assay, and 1.75 μM in the β-arrestin assay, and EC80 of 10 nM in both assays.

Smiles

[O-][N+](=O)c1ccc(cc1)C(=O)Oc1coc(CSc2ncccn2)cc1=O

Molecular Formula

C17H11N3O6S

Molecular Weight

385.35

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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