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GNE-617

Product Specifications

CAS Number

1362154-70-8

Target

NAMPT

Related Pathways

Metabolism

Purity

0.9997

Bioactivity

GNE-617, a specific NAMPT inhibitor (IC50=5 nM), shows potency in xenograft models of cancer.

Smiles

Fc1cc(F)cc(c1)S(=O)(=O)c1ccc(CNC(=O)c2ccc3nccn3c2)cc1

Molecular Formula

C21H15F2N3O3S

Molecular Weight

427.42

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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