GNE-617
Product Specifications
CAS Number
1362154-70-8
Target
NAMPT
Related Pathways
Metabolism
Purity
0.9997
Bioactivity
GNE-617, a specific NAMPT inhibitor (IC50=5 nM), shows potency in xenograft models of cancer.
Smiles
Fc1cc(F)cc(c1)S(=O)(=O)c1ccc(CNC(=O)c2ccc3nccn3c2)cc1
Molecular Formula
C21H15F2N3O3S
Molecular Weight
427.42
Shipping Conditions
Cool pack
Storage Temperature
-20°C
Available Sizes
Curated Selection
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