PF 429242
Product Specifications
CAS Number
947303-87-9
Target
Fatty Acid Synthase, Lipid, Virus Protease, NPC1L1
Related Pathways
Microbiology/Virology, Metabolism, Membrane transporter/Ion channel
Purity
0.9927
Bioactivity
PF-429242 is a competitive inhibitor of sterol regulatory element-binding protein (SREBP) site 1 protease (IC50 = 0.175 μM) . It is selective for site 1 protease against a panel of serine proteases. PF-429242 inhibits rate of cholesterol synthesis in CHO cells (IC50 = 0.53 μM) .
Smiles
N(C(=O)C1=CC=C(CN(CC)CC)C=C1)(CCC2=C(OC)C=CC=C2)[C@@H]3CCNC3
Molecular Formula
C25H35N3O2
Molecular Weight
409.56
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog
127669-ML550 100 µL
GUCA1C (GCAP3, Guanylyl Cyclase-activating Protein 3, Guanylate Cyclase Activator 1C) (MaxLight 550)
Sign In for Pricing
View Details 
MBS9319603-01 48 Well
Human TBC1 domain family member 3B, TBC1D3B ELISA Kit
Sign In for Pricing
View Details MBS9319603-02 96 Well
Human TBC1 domain family member 3B, TBC1D3B ELISA Kit
Sign In for Pricing
View Details