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AM966

Product Specifications

CAS Number

1228690-19-4

Target

LPL Receptor, LPA Receptor

Related Pathways

GPCR/G Protein

Purity

0.9979

Bioactivity

AM966, a excellent affinity, specific, oral LPA1 (IC50=17 nM) antagonist, suppresses LPA-stimulated intracellular calcium release.

Smiles

C[C@@H](OC(=O)Nc1c(C)noc1-c1ccc(cc1)-c1ccc(CC(O)=O)cc1)c1ccccc1Cl

Molecular Formula

C27H23ClN2O5

Molecular Weight

490.93

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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