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MS049 dihydrochloride

Product Specifications

CAS Number

2095432-59-8

Target

Histone Methyltransferase

Related Pathways

Chromatin/Epigenetic

Bioactivity

MS049 dihydrochloride is a selective and cell-active dual inhibitor of PRMT4 and PRMT6 (IC50=34/43 nM), capable of reducing Med12me2a and H3R2me2a levels in HEK293 cells.

Smiles

CNCCN(CC1)CCC1OCC2=CC=CC=C2.Cl.Cl

Molecular Formula

C15H26Cl2N2O

Molecular Weight

321.29

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

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