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MLS-0437605

Product Specifications

CAS Number

862975-18-6

Target

Phosphatase, Others

Related Pathways

Others, Metabolism

Bioactivity

MLS-0437605 is a potent and selective inhibitor of dual-specificity phosphatase 3 (DUSP3), with an IC50 of 3.7 μM. It exhibits higher selectivity towards DUSP3 in comparison to DUSP22 and other protein tyrosine phosphatases (PTPs) .

Smiles

COc1ccc(cc1)-c1nnc(Nc2nc3c(F)cccc3s2)o1

Molecular Formula

C16H11FN4O2S

Molecular Weight

342.35

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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