Sulfatinib
Product Specifications
CAS Number
1308672-74-3
Target
Potassium Channel|||VEGFR|||FGFR
Related Pathways
Membrane transporter/Ion channel|||Angiogenesis|||Tyrosine Kinase/Adaptors
Purity
>99.99%
Bioactivity
Sulfatinib (KDR-IN-1) (HMPL-012) is a potent and highly selective tyrosine kinase inhibitor against VEGFR1/2/3, FGFR1 and CSF1R with IC 50 s ranging from 1 to 24 nM.
Smiles
CN(C)CCNS(=O)(=O)Cc1cccc(Nc2nccc(Oc3ccc4[nH]c(C)cc4c3)n2)c1
Molecular Formula
C24H28N6O3S
Molecular Weight
480.58
Shipping Conditions
Cool pack
Storage Temperature
-20°C
Available Sizes
Curated Selection
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