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Sulfatinib

Product Specifications

CAS Number

1308672-74-3

Target

Potassium Channel, VEGFR, FGFR

Related Pathways

Membrane transporter/Ion channel, Angiogenesis, Tyrosine Kinase/Adaptors

Purity

>99.99%

Bioactivity

Sulfatinib (KDR-IN-1) (HMPL-012) is a potent and highly selective tyrosine kinase inhibitor against VEGFR1/2/3, FGFR1 and CSF1R with IC 50 s ranging from 1 to 24 nM.

Smiles

CN(C)CCNS(=O)(=O)Cc1cccc(Nc2nccc(Oc3ccc4[nH]c(C)cc4c3)n2)c1

Molecular Formula

C24H28N6O3S

Molecular Weight

480.58

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

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