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ETC-159

Product Specifications

CAS Number

1638250-96-0

Target

Porcupine, Wnt/beta-catenin

Related Pathways

Cytoskeletal Signaling, Stem Cells

Purity

0.994

Bioactivity

ETC-159 (ETC-1922159) is a potent, orally available PORCN inhibitor that inhibits β-catenin reporter activity with an IC50 of 2.9 nM.

Smiles

Cn1c2ncn(CC(=O)Nc3ccc(nn3)-c3ccccc3)c2c(=O)n(C)c1=O

Molecular Formula

C19H17N7O3

Molecular Weight

391.38

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

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