ETC-159
Product Specifications
CAS Number
1638250-96-0
Target
Porcupine, Wnt/beta-catenin
Related Pathways
Cytoskeletal Signaling, Stem Cells
Purity
0.994
Bioactivity
ETC-159 (ETC-1922159) is a potent, orally available PORCN inhibitor that inhibits β-catenin reporter activity with an IC50 of 2.9 nM.
Smiles
Cn1c2ncn(CC(=O)Nc3ccc(nn3)-c3ccccc3)c2c(=O)n(C)c1=O
Molecular Formula
C19H17N7O3
Molecular Weight
391.38
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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