CDK7/9-IN-1
Product Specifications
CAS Number
2747919-19-1
Target
Others, CDK
Related Pathways
Cell Cycle/Checkpoint, Others
Bioactivity
CDK7/9-IN-1 is a specific inhibitor of cyclin-dependent kinases 7/9 (CDK7/9), targeting CDK7 with IC50 values of 0.0656 μM without pre-incubation and 0.00574 μM after 3 hours pre-incubation, and displaying inhibitory activity against CDK9 with an IC50 of 2.14 μM after 3 hours pre-incubation, making it valuable for cancer research.
Smiles
CC(C)c1cnc2c(NC3CCN(C[C@@H]4CN(CCO4)C(=O)C=C)CC3)cc(cn12)C(F)(F)F
Molecular Formula
C24H32F3N5O2
Molecular Weight
479.548
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
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