EPZ-719
Product Specifications
CAS Number
2697176-16-0
Target
Histone Methyltransferase, Others
Related Pathways
Chromatin/Epigenetic, Others
Bioactivity
EPZ-719 is a highly selective and potent inhibitor of SETD2, a novel compound known for its ability to inhibit the enzymatic activity of SETD2 (IC50 = 0.005 μM) . This compound displays a remarkable selectivity over other histone methyltransferases, making it a promising candidate for targeted therapeutic applications in the field of epigenetic research.
Smiles
CN([C@H]1CCN(C1)[C@H]1CCC[C@H](C1)NC(=O)c1cc2c(F)ccc(C)c2[nH]1)S(C)(=O)=O
Molecular Formula
C22H31FN4O3S
Molecular Weight
450.57
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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