OM99-2 TFA

Product Specifications

CAS Number

2504147-81-1

Target

Beta-Secretase

Related Pathways

Neuroscience

Bioactivity

OM99-2 TFA is an eight-residue peptidomimetic compound, functioning as a tight-binding inhibitor of human brain memapsin 2. It exhibits a high affinity for the target with a Ki value of 9.58 nM, making it a promising candidate in the development of BACE1 inhibitors. Due to its potential, OM99-2 presents opportunities for further research in the field of Alzheimer's disease.

Smiles

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