FTX-6058
Product Specifications
CAS Number
2490676-18-9
Target
Histone Methyltransferase, Others
Related Pathways
Others, Chromatin/Epigenetic
Bioactivity
FTX-6058 is a potent orally active inhibitor targeting Embryonic Ectoderm Development (EED) . It effectively induces HbF protein expression in both cell and murine models. This compound holds significant potential for researching select hemoglobinopathies such as sickle cell disease and β-thalassemia.
Smiles
Cc1ncccc1-c1cc2OC[C@H]3COc4ccc(F)c(CNc2n2cnnc12)c34
Molecular Formula
C22H18FN5O2
Molecular Weight
403.417
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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