What is the catalog number for MS67?

The catalog number for MS67 is T39976.

What sizes are available for MS67?

MS67 is available in the following size(s): 10 mg.

MS67 is currently made to order / not held in immediate stock. Contact us for lead time.

Who manufactures MS67?

MS67 is manufactured by Molfinity.

What is the estimated delivery time for MS67?

Estimated delivery time for MS67 is approximately 10 business day(s), depending on your location.

MS67

Product Specifications

CAS Number

2407452-77-9

Target

PROTACs, Histone Methyltransferase

Related Pathways

PROTAC, Chromatin/Epigenetic

Bioactivity

MS67 is a potent and selective degrader of WD40 repeat domain protein 5 (WDR5) with a dissociation constant (Kd) of 63 nM, exhibiting no activity against protein methyltransferases, kinases, G-protein-coupled receptors (GPCRs), ion channels, and transporters, and notably demonstrating significant anticancer properties.

Smiles

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