M-808
Product Specifications
CAS Number
2377335-74-3
Target
Others, Epigenetic Reader Domain
Related Pathways
Chromatin/Epigenetic, Others
Bioactivity
M-808 is a potent and efficacious covalent inhibitor, targeting the interaction between Menin and MLL. It demonstrates a high binding affinity with an IC50 value of 2.6 nM.
Smiles
[H][C@@]1(CCC[C@@H]1NC(=O)OC)[C@@](CN1CCC1)(C1CCN(CC2CN(C2)c2ccc(cc2)S(=O)(=O)C2CN(C2)C(=O)\C=C\CN2CCCCC2)CC1)c1cccc(F)c1
Molecular Formula
C45H63FN6O5S
Molecular Weight
819.09
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Frequently Asked Questions
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