TBK1/IKKε-IN-6
Product Specifications
CAS Number
2306877-20-1
Target
IκB/IKK, Others
Related Pathways
Others, NF-κB
Bioactivity
TBK1/IKKε-IN-6 (example 110) is a potent inhibitor of TBK1 and IKKε, exhibiting IC50 values below 100 nM for both enzymes.
Smiles
COc1nc(Nc2nccc(n2)-c2ccc(OC3CCN(CC3(F)F)C(=O)[C@@H](C)O)c(c2)C#N)ccc1N1CCN(C)C[C@H]1C
Molecular Formula
C31H36F2N8O4
Molecular Weight
622.678
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Frequently Asked Questions
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