BRK inhibitor P21d hydrochloride
Product Specifications
CAS Number
2250025-98-8
Target
Others, BTK
Related Pathways
Tyrosine Kinase/Adaptors, Angiogenesis, Others
Bioactivity
BRK inhibitor P21d hydrochloride is a highly potent inhibitor of breast tumor kinase (BRK/PTK6), displaying an IC50 of 30 nM, and effectively suppresses p-SAM68 with an IC50 of 52 nM. This compound serves as a valuable tool for evaluating BRK inhibitors' efficacy in xenograft breast tumor models, enabling in vivo activity assessment.
Smiles
Cl.Fc1cc(ccc1Nc1nc(cn2c(cnc12)-c1cn[nH]c1)C1CC1)C(=O)N1CCOCC1
Molecular Formula
C23H23ClFN7O2
Molecular Weight
483.93
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
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