ERα degrader-2
Product Specifications
CAS Number
2235396-63-9
Target
ERK, Estrogen Receptor/ERR
Related Pathways
Endocrinology/Hormones, MAPK
Purity
0.9971
Bioactivity
ERα degrader-2 is a selective and potent estrogen receptor (SERD) degrader with anticancer activity, exhibiting an EC50 value of 0.3 nM for ERα degradation. It can be used for the prevention and treatment of HER-positive breast cancer.
Smiles
[H][C@@]1(N(CC(C)(C)F)[C@H](C)Cc2c1[nH]c1ccccc21)c1c(F)cc(cc1F)-c1ccc(cc1)C(O)=O
Molecular Formula
C29H27F3N2O2
Molecular Weight
492.53
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
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