BMS-986278
Product Specifications
CAS Number
2170126-74-4
Target
LPA Receptor, LPL Receptor
Related Pathways
GPCR/G Protein
Purity
0.9988
Bioactivity
BMS-986278 is an orally active and potent hemophosphatidic acid receptor 1 (LPA1) antagonist with Kb values of 6.9 nM and 4.0 nM for human and mouse LPA1, respectively.BMS-986278 may be investigated for use in idiopathic pulmonary fibrosis.
Smiles
CCCN(C)C(=O)OCc1c(nnn1C)-c1ccc(O[C@H]2CCC[C@@H](C2)C(O)=O)c(C)n1
Molecular Formula
C22H31N5O5
Molecular Weight
445.51
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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