GSK097
Product Specifications
CAS Number
2159137-02-5
Target
Epigenetic Reader Domain, Others
Related Pathways
Others, Chromatin/Epigenetic
Bioactivity
GSK097 is a highly potent and selective inhibitor of the second bromodomain (BD2) found in bromodomain and extra-terminal domain (BET) proteins. It exhibits a remarkable 2000-fold selectivity for BD2 over BD1, as indicated by BRD4 data. Additionally, GSK097 demonstrates solubility of over 1 mg/mL in FaSSIF media.
Smiles
CNC(=O)c1cc(cc(n1)[C@@H](O)c1ccccc1)C(=O)N[C@H]1C[C@@H]1C
Molecular Formula
C19H21N3O3
Molecular Weight
339.395
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Frequently Asked Questions
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