Apalutamide-COOH
Product Specifications
CAS Number
1332391-04-4
Target
Others, Drug Metabolite
Related Pathways
Others, Metabolism
Bioactivity
Apalutamide-COOH is a metabolite derived from Apalutamide, which acts as a highly potent and competitive antagonist of the androgen receptor (AR) . It effectively binds to the AR with an IC50 value of 16 nM.
Smiles
OC(=O)c1ccc(cc1F)N1C(=S)N(C(=O)C11CCC1)c1cnc(C#N)c(c1)C(F)(F)F
Molecular Formula
C20H12F4N4O3S
Molecular Weight
464.39
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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