Ro 1138452 hydrochloride
Product Specifications
Target
Others
Related Pathways
Others
Bioactivity
Selective prostacyclin IP receptor antagonist (pKi = 8.3) . Exhibits no affinity at other prostanoid receptors (EP1-4, FP and TP) in a radioligand binding assay. Demonstrates analgesic activity in rats. Orally bioavailable.
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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