(R) -KT109
Product Specifications
CAS Number
2055172-60-4
Target
Others
Related Pathways
Others
Bioactivity
(R) -KT109 is the (R) isomer of the diacylglycerol lipase β (DAGLβ) inhibitor KT109 . (R) -KT109 is an inhibitor of DAGLβ (IC50 = 0.79 nM) and of DAGLα-mediated hydrolysis of 1-stearoyl-2-arachidonoyl-sn-glycerol . It also inhibits α/β-hydrolase domain-containing protein 6 (ABHD6) with an IC50 value of 2.51 nM. (R) -KT109 is more potent at DAGLβ, DAGLα, and ABHD6 than (S) -KT109 .
Smiles
C(=O)(N1[C@@H](CC2=CC=CC=C2)CCCC1)N3C=C(N=N3)C4=CC=C(C=C4)C5=CC=CC=C5
Molecular Formula
C27H26N4O
Molecular Weight
422.52
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog
036201-ML490 100 µL
GPHN, ID (GPHN, GPH, KIAA1385, Gephyrin, Molybdopterin adenylyltransferase, Domain G, Molybdopterin molybdenumtransferase, Domain E) (MaxLight 490) discontinued
Sign In for Pricing
View Details