Bilaid C
Product Specifications
CAS Number
2393866-13-0
Target
Opioid Receptor
Related Pathways
Neuroscience, Endocrinology/Hormones, GPCR/G Protein
Bioactivity
Bilaid C is a tetrapeptide μ-opioid receptor agonist (Ki= 210 nM in HEK293 cell membranes expressing the human receptor) that has been found inPenicillium.1It inhibits forskolin-induced cAMP accumulation by 77% in HEK293 cells expressing the human μ-opioid receptor when used at a concentration of 10 μM. Bilaid C induces inward rectifying potassium channel (Kir) currents in rat locus coeruleus slices that endogenously express high levels of the μ-opioid receptor (EC50= 4.2 μM) .
Smiles
CC(C)[C@H](NC(=O)[C@H](NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(C)C)C(=O)N[C@H](Cc1ccccc1)C(O)=O
Molecular Formula
C28H38N4O6
Molecular Weight
526.62
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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