CB2R PAM
Product Specifications
CAS Number
2244579-87-9
Target
Cannabinoid Receptor
Related Pathways
GPCR/G Protein
Purity
0.9909
Bioactivity
CB2R PAM is an orally active cannabinoid type 2 receptor (CB2Rs) positive allosteric modulator that enhances CP 55940 and 2-Arachidonylglycerol-stimulated [35S]GTP?S binding to CB2 receptors without affecting receptor activity in the absence of agonists. CB2R PAM shows anti-injury activity in a mouse model of neuropathic pain.
Smiles
N(C(=O)C1CCCCCC1)C=2C(=O)N(CC3=CC=C(F)C=C3)C=C(Br)C2C
Molecular Formula
C21H24BrFN2O2
Molecular Weight
435.33
Shipping Conditions
Cool pack
Storage Temperature
-20°C
Available Sizes
Curated Selection
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