Cutamesine
Product Specifications
CAS Number
165377-43-5
Target
Sigma receptor
Related Pathways
GPCR/G Protein
Bioactivity
Cutamesine (SA4503; AGY-94806), a selective sigma 1 receptor (σ1R) agonist, exhibits high affinity for the σ1R subtype as indicated by (+) -[3H]pentazocine labeling, with an IC50 value of 17.4±1.9 nM. It demonstrates 100-fold lower affinity for the sigma 2 receptor.
Smiles
COc1ccc(CCN2CCN(CCCc3ccccc3)CC2)cc1OC
Molecular Formula
C23H32N2O2
Molecular Weight
368.51
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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