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PDE4B-IN-2

Product Specifications

CAS Number

915082-52-9

Target

PDE

Related Pathways

Metabolism

Purity

0.9937

Bioactivity

PDE4B-IN-2 (A 33) is an orally active and selective PDE4B inhibitor with an IC50 of 15 nM. PDE4B-IN-2 inhibits PDE4D (IC50=1.7 μM) . PDE4B-IN-2 exhibits potent anti-inflammatory effects.

Smiles

CCc1c(C)nc(nc1Nc1ccc(CC(O)=O)cc1)-c1ccc(Cl)s1

Molecular Formula

C19H18ClN3O2S

Molecular Weight

387.88

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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