PDE4B-IN-2
Product Specifications
CAS Number
915082-52-9
Target
PDE
Related Pathways
Metabolism
Purity
0.9937
Bioactivity
PDE4B-IN-2 (A 33) is an orally active and selective PDE4B inhibitor with an IC50 of 15 nM. PDE4B-IN-2 inhibits PDE4D (IC50=1.7 μM) . PDE4B-IN-2 exhibits potent anti-inflammatory effects.
Smiles
CCc1c(C)nc(nc1Nc1ccc(CC(O)=O)cc1)-c1ccc(Cl)s1
Molecular Formula
C19H18ClN3O2S
Molecular Weight
387.88
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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