UPSEM 817 tartrate
Product Specifications
CAS Number
2341833-14-3
Target
Others
Related Pathways
Others
Bioactivity
Selective ultrapotent PSEM (uPSEM) agonist for α7L131G, Q139L, Y217F-GlyR (PSAM4-GlyR) and PSAM4-5-HT3 chimeric ion channel agonist (EC50 values are 0.3 and 0.5 nM, respectively) . Suppresses firing of layer 2/3 cortical neurons expressing PSAM4-GlyR in brain slices. Increases contralateral rotation in mice expressing PSAM4-GlyR unilaterally in the substantia nigra reticulata (LED 0.1 mg/kg) .
Smiles
O[C@H]([C@@H](O)C(O)=O)C(O)=O.CCCOc1cnc2cc3C4CC(CNC4)c3cc2n1 |THB:27:26:21:23.24.25,18:19:21:23.24.25|
Molecular Formula
C20H25N3O7
Molecular Weight
419.434
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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