Rupatadine
Product Specifications
CAS Number
158876-82-5
Target
Histamine Receptor, Autophagy, PAFR
Related Pathways
Neuroscience, Autophagy, GPCR/G Protein, Immunology/Inflammation
Purity
0.9987
Bioactivity
Rupatadine (UR-12592, rupatadine) is a potent and orally available dual antagonist of PAF and histamine H1 receptors with Ki values of 0.55 μM and 0.1 μM, respectively, which provides relief of allergic symptoms and anti-inflammatory properties, and is used in allergic rhinitis and chronic urticaria.
Smiles
ClC=1C=CC2=C(C1)CCC=3C=CC=NC3C2=C4CCN(CC=5C=NC=C(C5)C)CC4
Molecular Formula
C26H26ClN3
Molecular Weight
415.96
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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