What is the catalog number for Relugolix?

The catalog number for Relugolix is T3630.

What sizes are available for Relugolix?

Relugolix is available in the following size(s): 2 mg, 5 mg, 1 mL - 10 mM (in DMSO), 10 mg, 25 mg, 50 mg, 100 mg, 200 mg.

How many pack sizes does Relugolix come in?

Relugolix is available in 8 different pack sizes.

Is Relugolix in stock?

Relugolix is currently made to order / not held in immediate stock. Contact us for lead time.

Who manufactures Relugolix?

Relugolix is manufactured by Molfinity.

What is the estimated delivery time for Relugolix?

Estimated delivery time for Relugolix is approximately 10 business day(s), depending on your location.

Relugolix

Product Specifications

CAS Number

737789-87-6

Target

GNRH Receptor

Related Pathways

GPCR/G Protein

Purity

0.9997

Bioactivity

Relugolix (RVT-601) is an orally available, non-peptide gonadotropin-releasing hormone (GnRH or luteinizing hormone-releasing hormone (LHRH) ) antagonist, with potential antineoplastic activity. Relugolix competitively binds to and blocks the GnRH receptor in the anterior pituitary gland, which both prevents GnRH binding to the GnRH receptor and inhibits the secretion and release of both luteinizing hormone (LH) and follicle stimulating hormone (FSH) . In males, the inhibition of LH secretion prevents the release of testosterone from Leydig cells in the testes. Since testosterone is required to sustain prostate growth, reducing testosterone levels may inhibit hormone-dependent prostate cancer cell proliferation.