(E/Z) -THZ1 2HCl
Product Specifications
CAS Number
2095433-94-4
Target
CDK
Related Pathways
Cell Cycle/Checkpoint
Purity
0.9951
Bioactivity
THZ1 2HCl (THZ1 Dihydrochloride) is a selective, covalent, and allosteric inhibitor of CDK7 with an IC50 of 3.2 nM. THZ1 2HCl has antiproliferative effects on a variety of cancer cell lines.
Smiles
Cl.Cl.CN(C)C\C=C\C(=O)Nc1ccc(cc1)C(=O)Nc1cccc(Nc2ncc(Cl)c(n2)-c2c[nH]c3ccccc23)c1
Molecular Formula
C31H30Cl3N7O2
Molecular Weight
638.98
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog
MBS1255071-01 0.02 mg (E-Coli)
Recombinant Shewanella sp. 3,4-dihydroxy-2-butanone 4-phosphate synthase (ribB)
Sign In for Pricing
View Details MBS1255071-02 0.1 mg (E-Coli)
Recombinant Shewanella sp. 3,4-dihydroxy-2-butanone 4-phosphate synthase (ribB)
Sign In for Pricing
View Details MBS1255071-03 0.02 mg (Yeast)
Recombinant Shewanella sp. 3,4-dihydroxy-2-butanone 4-phosphate synthase (ribB)
Sign In for Pricing
View Details MBS1255071-04 0.1 mg (Yeast)
Recombinant Shewanella sp. 3,4-dihydroxy-2-butanone 4-phosphate synthase (ribB)
Sign In for Pricing
View Details