Relamorelin
Product Specifications
CAS Number
661472-41-9
Target
GHSR
Related Pathways
GPCR/G Protein
Purity
>99.99%
Bioactivity
Relamorelin (BIM28131, RM131) is a selective and potent ghrelin/growth hormone secretagogue receptor (GHSR) agonist with high affinity for GHS-1a receptor (Ki value is 0.42 ± 0.063 nM) . Relamorelin (BIM28131, RM131) is also a centrally permeable pentapeptide analog that can increase growth hormone levels and accelerate gastric emptying, and has the potential to study cachexia.
Smiles
C([C@@H](NC([C@@H](CC=1C=2C(SC1)=CC=CC2)NC(=O)C3CCNCC3)=O)C(N[C@H](C(NC4(C(N)=O)CCNCC4)=O)CC5=CC=CC=C5)=O)C=6C=7C(NC6)=CC=CC7
Molecular Formula
C43H50N8O5S
Molecular Weight
790.97
Shipping Conditions
Ice Packs
Storage Temperature
-20°C