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AKT inhibitor VIII

Product Specifications

CAS Number

612847-09-3

Target

Apoptosis, Akt

Related Pathways

PI3K/Akt/mTOR signaling, Cytoskeletal Signaling, Apoptosis

Purity

0.9877

Bioactivity

AKT inhibitor VIII (AKTi-1/2) is a highly specific inhibitor of Akt1/2, with IC50 values of 58 nM and 210 nM respectively, demonstrating approximately 36-fold greater selectivity for Akt1 over Akt3.

Smiles

O=c1[nH]c2ccccc2n1C1CCN(Cc2ccc(cc2)-c2nc3cc4[nH]cnc4cc3nc2-c2ccccc2)CC1

Molecular Formula

C34H29N7O

Molecular Weight

551.64

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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