Ecopipam
Product Specifications
CAS Number
112108-01-7
Target
5-HT Receptor, Dopamine Receptor, Adrenergic Receptor
Related Pathways
GPCR/G Protein, Neuroscience
Purity
0.9968
Bioactivity
Ecopipam (UNII-0X748O646K) is a potent, selective, and orally active antagonist of dopamine D1/D5 receptors, with Kis of 1.2 nM and 2.0 nM, respectively. Ecopipam demonstrates more than 40-fold selectivity over D2, D4, 5-HT, and α2a receptors (Ki=0.98, 5.52, 0.08, and 0.73 μM, respectively) . It is used in research on schizophrenia and obesity.
Smiles
CN1[C@@]2([C@@](C=3C(=CC(Cl)=C(O)C3)CC1)(C=4C(CC2)=CC=CC4)[H])[H]
Molecular Formula
C19H20ClNO
Molecular Weight
313.82
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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