CP 461
Product Specifications
CAS Number
227619-96-7
Target
PDE, Microtubule Associated, Apoptosis
Related Pathways
Metabolism, Cytoskeletal Signaling, Apoptosis
Purity
0.9982
Bioactivity
CP 461 (UNII-68OJX9I7DT), a specific PDE2A inhibitor, is a novel pro-apoptotic compound that inhibits cyclic GMP phosphodiesterase but not cyclooxygenase-1 or -2. CP 461 inhibits the growth of a variety of human tumor cell lines in vitro and selectively induces apoptosis in cancer cell lines, but not in normal cells.
Smiles
C(C(NCC1=CC=CC=C1)=O)C=2C=3C(/C(=C\C=4C=CN=CC4)/C2C)=CC=C(F)C3.Cl
Molecular Formula
C25H22ClFN2O
Molecular Weight
420.91
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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