Cerlapirdine
Product Specifications
CAS Number
925448-93-7
Target
5-HT Receptor
Related Pathways
GPCR/G Protein, Neuroscience
Purity
0.9877
Bioactivity
Cerlapirdine (PF-05212365) is a selective, potent, full antagonist of the 5-hydroxytryptamine 6 (5-HT6) receptor. Cerlapirdine is already in clinical development for the treatment of cognitive disorders related to Alzheimer's disease and schizophrenia. It works by acting as a selective 5-HT6 receptor antagonist.
Smiles
S(=O)(=O)(C=1C=2C(NN1)=CC=C(OCCCN(C)C)C2)C=3C4=C(C=CC3)C=CC=C4
Molecular Formula
C22H23N3O3S
Molecular Weight
409.5
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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