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PF-670462

Product Specifications

CAS Number

950912-80-8

Target

Casein Kinase

Related Pathways

Metabolism, Stem Cells

Purity

0.9972

Bioactivity

PF-670462 is a potent (IC50 = 7.7 ± 2.2 nM) and selective (>30-fold with respect to 42 additional kinases) inhibitor of CK1ε in isolated enzyme preparations.

Smiles

Cl.Cl.Nc1nccc(n1)-c1c(ncn1C1CCCCC1)-c1ccc(F)cc1

Molecular Formula

C19H22Cl2FN5

Molecular Weight

410.32

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

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