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VU0477886

Product Specifications

CAS Number

1926222-30-1

Target

GluR, Others

Related Pathways

Others, Neuroscience

Bioactivity

VU0477886 is a potent mGlu4 positive allosteric modulator (PAM) with robust efficacy in a standard preclinical Parkinson's disease model, haloperidol-induced catalepsy (HIC) .

Smiles

O=C(C1=NC=CC=C1N)NC2=CC=C(N(C(C3=C4C=CC=C3)=O)C4=O)C(Cl)=C2

Molecular Formula

C20H13ClN4O3

Molecular Weight

392.8

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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